Binding to an unusual inactive kinase conformation by highly selective to inhibitors of inositol-requiring enzyme 1ɑ kinase-endoribonuclease

Giampiero Colombano, John J. Caldwell, Thomas P. Matthews, Chitra Bhatia, Amar Joshi, Tatiana McHardy, Ngai Yi Mok, Yvette Newbatt, Lisa Pickard, Jade Strover, Somaieh Hedayat, Michael I. Walton, Stephanie M. Myers, Alan M. Jones, Harry Saville, Craig McAndrew, Rosemary Burke, Suzanne A. Eccles, Faith E. Davies, Richard BaylissIan Collins

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Medicine & Life Sciences

Chemistry