Journal of Medicinal Chemistry, 0022-2623
Journal
Publications
- 2021
- E-pub ahead of print
Discovery of Novel Thiophene-arylamide Derivatives as DprE1 Inhibitors with Potent Antimycobacterial Activities
Sarah Batt, Del Besra, 14 Apr 2021, In: Journal of Medicinal Chemistry.Research output: Contribution to journal › Article › peer-review
- 2020
- E-pub ahead of print
Discovery of highly selective inhibitors of calmodulin-dependent kinases that restore insulin sensitivity in the diet-induced obese in vivo mouse model
Graziella Greco, Marc Lenoir, Clare Box, Vera Novitskaya & 14 others, , 20 May 2020, In: Journal of Medicinal Chemistry.Research output: Contribution to journal › Article › peer-review
- Published
Investigation of inactive state κ opioid receptor homodimerization via single molecule microscopy using new antagonistic fluorescent probes
Zsombor Koszegi, Yann Lanoiselee, Davide Calebiro, 9 Apr 2020, In: Journal of Medicinal Chemistry. 63, 7, p. 3596-3609 14 p.Research output: Contribution to journal › Article › peer-review
- 2019
- Published
Design, synthesis and biological evaluation of a new series of carvedilol derivatives that protect sensory hair cells from aminoglycoside-induced damage by blocking the mechano-electrical transducer channel
Molly O'Reilly, 13 Jun 2019, In: Journal of Medicinal Chemistry. 62, 11, p. 5312-5329 18 p.Research output: Contribution to journal › Article › peer-review
- Published
Binding to an unusual inactive kinase conformation by highly selective to inhibitors of inositol-requiring enzyme 1ɑ kinase-endoribonuclease
Alan M Jones & 1 others, , 1 Mar 2019, In: Journal of Medicinal Chemistry. 62, 5, p. 2447-2465 19 p.Research output: Contribution to journal › Article › peer-review
- 2018
- Published
In vivo selectivity and localization of reactive oxygen species (ROS) induction by osmium anticancer complexes that circumvent platinum resistance
Isolda Romero-Canelón, 25 Oct 2018, In: Journal of Medicinal Chemistry. 61, 20, p. 9246–9255 10 p.Research output: Contribution to journal › Article › peer-review
- Published
Targeting multiple effector pathways in pancreatic ductal adenocarcinoma with a g-quadruplex-binding small molecule
Jeremy Pike & 3 others, , 22 Mar 2018, In: Journal of Medicinal Chemistry. 61, 6, p. 2500-2517 18 p.Research output: Contribution to journal › Article › peer-review
- Published
Synthesis and Biological Evaluation of (E)-4-Hydroxy-3-Methylbut-2-enyl Phosphate (HMBP) Aryloxy Triester Phosphoramidate Prodrugs as Activators of Vγ9/Vδ2 T-Cells Immune Response
Martin Davey, Taher Taher, Benjamin Willcox & Youcef Mehellou, 19 Feb 2018, In: Journal of Medicinal Chemistry. 61, 5, p. 2111-2117Research output: Contribution to journal › Article › peer-review
- Published
BACE-1 Inhibitors: From Recent Single-Target Molecules to Multitarget Compounds for Alzheimer's Disease
Giovanni Bottegoni, 8 Feb 2018, In: Journal of Medicinal Chemistry. 61, 3, p. 619-637 19 p.Research output: Contribution to journal › Review article › peer-review
- 2017
- E-pub ahead of print
Quinazolinone-based Anticancer Agents: Synthesis, Anti-proliferative SAR, Anti-tubulin Activity and Tubulin Co-crystal Structure
Paul Foster, 11 Dec 2017, In: Journal of Medicinal Chemistry.Research output: Contribution to journal › Article › peer-review