1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman; Joshua D. Tibbetts; Steven D. Bull

doi:10.1016/j.tet.2018.05.044

1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman, Joshua D. Tibbetts, Steven D. Bull

Chemistry

Research output: Contribution to journal › Article › peer-review

Abstract

1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

Original language	English
Pages (from-to)	5330-5339
Number of pages	10
Journal	Tetrahedron
Volume	74
Issue number	38
DOIs	https://doi.org/10.1016/j.tet.2018.05.044
Publication status	Published - 20 Sept 2018

Keywords

1
1-Acylals
Amides
N-Acylation
Solvent free

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10.1016/j.tet.2018.05.044

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title = "1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines",

abstract = "1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.",

keywords = "1, 1-Acylals, Amides, N-Acylation, Solvent free",

author = "Chapman, {Robert S.L.} and Tibbetts, {Joshua D.} and Bull, {Steven D.}",

year = "2018",

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T1 - 1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

AU - Chapman, Robert S.L.

AU - Tibbetts, Joshua D.

AU - Bull, Steven D.

PY - 2018/9/20

Y1 - 2018/9/20

N2 - 1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

AB - 1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

KW - 1

KW - 1-Acylals

KW - Amides

KW - N-Acylation

KW - Solvent free

U2 - 10.1016/j.tet.2018.05.044

DO - 10.1016/j.tet.2018.05.044

M3 - Article

SN - 0040-4020

VL - 74

SP - 5330

EP - 5339

JO - Tetrahedron

JF - Tetrahedron

IS - 38

ER -

1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Abstract

Keywords

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