MICA: Addressing the burgeoning problem of tuberculosis: Exploiting phenotypic hits to identify new protein targets for drug discovery

Short title	MICA: Addressing the burgeoning problem of tuberculosis: Exploiting phenotypic hits to identify new protein targets for drug discovery
Status	Finished
Effective start/end date	1/04/18 → 31/03/22

Exploration of vanoxerine analogues as antibacterial agents
Kingdon, A. D. H., Adcock, H. V., Kasimati, E.-M., Craven, P., van Schaik, W., Cox, L. R. & Besra, G. S., Jan 2025, In: The Journal of antibiotics. 78, 1, p. 54-63 10 p.
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The deacetylase NagA mediates the remodelling and recycling of peptidoglycan derived amino sugars in mycobacteria
Guy, C. S., Cooper, C., Karlikowska, M., Harrison, J., Singh, A., Servín-González, L. S., Evans, C. A., Bakker, S. E., Bottrill, A., Bhatt, A., Mesnage, S., Besra, G. S. & Fullam, E., 14 Aug 2025, (E-pub ahead of print) In: The Journal of biological chemistry. 110597.
Research output: Contribution to journal › Article › peer-review

Open Access
Novel hybrids of 1,2,3-triazole-benzoxazole: design, synthesis, and assessment of DprE1 enzyme inhibitors using fluorometric assay and computational analysis
Singh, M., Batt, S. M., Canales, C. S. C., Pavan, F. R., Kumar, S. A., Akshatha, H. S., Bhagyalalitha, M., Pujar, K. G., Bidye, D., Pujar, G. V. & Besra, G. S., 31 Dec 2024, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 39, 1, 16 p., 2403744.
Research output: Contribution to journal › Article › peer-review

Open Access
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